| 1 |
Apralogs: Apramycin 5-O-Glycosides and Ethers with Improved Antibacterial Activity and Ribosomal Selectivity and Reduced Susceptibility to the Aminoacyltranserferase (3)-IV Resistance Determinant
Quirke JCK, Rajasekaran P, Sarpe V, Sonousi A, Osinnii I, Gysin M, Haldimann K, Fang QJ, Shcherbakov D, Hobbie SN, Sha SH, Schacht J, Vasella A, Bottger EC, Crich D
Journal of the American Chemical Society, 142(1), 530, 2020 |
| 2 |
Design, Multigram Synthesis, and in Vitro and in Vivo Evaluation of Propylamycin: A Semisynthetic 4,5-Deoxystreptamine Class Aminoglycoside for the Treatment of Drug-Resistant Enterobacteriaceae and Other Gram-Negative Pathogens
Matsushita T, Sati GC, Kondasinghe N, Pirrone MG, Kato T, Waduge P, Kumar HS, Sanchon AC, Dobosz-Bartoszek M, Shcherbakov D, Juhas M, Hobbie SN, Schrepfer T, Chow CS, Polikanov YS, Schacht J, Vasella A, Bottger EC, Crich D
Journal of the American Chemical Society, 141(12), 5051, 2019 |
| 3 |
Solution chemistry of copper(II)-gentamicin complexes: Relevance to metal-related aminoglycoside toxicity
Lesniak W, Harris WR, Kravitz JY, Schacht J, Pecoraro VL
Inorganic Chemistry, 42(5), 1420, 2003 |
| 4 |
The molecular and crystal structures of three 4-(omega-cyanoalkyloxy)benzoic acids and of a 1 : 1 ordered mixed crystal of 4-(omega-cyanobutyloxy)benzoic acid and 4-(omega-cyanopentyloxy)benzoic acid formed by hydrogen bonding
Zugenmaier P, Bock I, Schacht J
Molecular Crystals and Liquid Crystals, 392, 31, 2002 |
