Chemistry Letters, Vol.33, No.5, 594-595, 2004
Useful method for direct introduction of the photoaffinity 3-(4-hydroxyphenyl)-3-trifluoromethyldiazirine group
A convergent and efficient preparation method of the photo-affinity 3-(4-alkoxyphenyl)-3-trifluoroinethyldiazirine derivatives was established by direct introduction of the photoaffinity group utilizing the Mitsunobu reaction.